2-(aminomethyl)pentan-1-ol

反応条件: temp:0.00; pressure:0.00; stir:; See reaction.notes.procedure_details.

実験手順: The title compound was synthesized in analogy to Example 102, using 5-bromo-6-hydroxy-nicotinic acid methyl ester, 2-methoxyethanol, (4-chloro-phenyl)-boronic acid and 2-(aminomethyl)-1-pentanol as starting materials to yield (RS)-5-(4-chloro-phenyl)-N-(2-hydroxymethyl-pentyl)-6-(2-methoxy-ethoxy)-nicotinamide. MS (ISP) 407.5 (M+H)+. The title compound was synthesized in analogy to Example 102